Invited Talk 21st International Conference on Biological Inorganic Chemistry 2025

How does haem alter the behaviour of the core clock proteins? (125575)

Andrew Hudson 1 , Kornelija Rimgailaite 1 , Mae James 1 , Christiane Reick 1 , Ezio Rosato 2 , Charalambos Kyriacou 2 , Emma Raven 3
  1. School of Chemistry, University of Leicester, Leicester
  2. Department of Genetics, Genomics and Cancer Sciences, University of Leicester, Leicester
  3. School of Chemistry, University of Bristol, Bristol

Thousands of different proteins are known, spanning the whole of the biological world, that contain haem as an integral component. Haemoproteins are responsible for binding and transportation of gaseous molecules, biochemical catalysis, and redox reactions in the electron-transport chain. Haem itself is a simple organo-transition-metal compound containing iron at the centre of a porphyrin macrocycle. By providing a metal centre for gas binding, substrate binding and charge transfer, haem is pivotal to the biochemical function of a haemoprotein. Traditionally, haem’s role was considered to be confined to haemoproteins with specific binding pockets, where it is a tightly bound and essential prosthetic group. Emerging evidence has dramatically shifted this view, revealing that haem also exists in an exchangeable pool within cells capable of transiently binding to a wider range of proteins, including those not classically defined as haemoproteins. cell.[1, 2]

We have been investigating how haem interacts with circadian-clock proteins in ways that impact their ability to form protein–protein or protein–DNA complexes. Specifically, we have been using NMR, fluorescence lifetime and correlation spectroscopy and light scattering techniques. In parallel, we have performed cellular assays to identify changes in circadian rhythmicity caused by excesses and deficiencies in haem.

 

  1. Leung, G.C., et al., Unravelling the mechanisms controlling heme supply and demand. Proc Natl Acad Sci U S A, 2021. 118(22).
  2. Gallio, A.E., et al., Understanding the Logistics for the Distribution of Heme in Cells. JACS Au, 2021. 1(10): p. 1541-1555.